Andexanet alfa for the reversal of Factor Xa inhibitor related anticoagulation

dc.contributor.author

Ghadimi, K

dc.contributor.author

Welsby, IJ

dc.contributor.author

Levy, JH

dc.contributor.author

Dombrowski, KE

dc.date.accessioned

2024-01-13T17:03:40Z

dc.date.available

2024-01-13T17:03:40Z

dc.date.issued

2016-01

dc.description.abstract

Andexanet alfa is a specific reversal agent for Factor Xa inhibitors. The molecule is a recombinant protein analog of factor Xa that binds to Factor Xa inhibitors and antithrombin:LMWH complex but does not trigger prothrombotic activity. In ex vivo, animal, and volunteer human studies, andexanet alfa (AnXa) was able to dose-dependently reverse Factor Xa inhibition and restore thrombin generation for the duration of drug administration. Further trials are underway to examine its safety and efficacy in the population of patients experiencing FXa inhibitor-related bleeding.

dc.identifier.issn

1747-4086

dc.identifier.issn

1747-4094

dc.identifier.uri

https://hdl.handle.net/10161/29789

dc.language

eng

dc.publisher

Informa UK Limited

dc.relation.ispartof

Expert review of hematology

dc.relation.isversionof

10.1586/17474086.2016.1135046

dc.rights.uri

https://creativecommons.org/licenses/by-nc/4.0

dc.subject

Animals

dc.subject

Humans

dc.subject

Factor Xa

dc.subject

Recombinant Proteins

dc.subject

Drug Evaluation, Preclinical

dc.subject

Protein Binding

dc.subject

Blood Coagulation

dc.subject

Clinical Trials, Phase I as Topic

dc.subject

Clinical Trials, Phase II as Topic

dc.subject

Clinical Trials, Phase III as Topic

dc.subject

Factor Xa Inhibitors

dc.title

Andexanet alfa for the reversal of Factor Xa inhibitor related anticoagulation

dc.type

Journal article

duke.contributor.orcid

Ghadimi, K|0000-0002-9287-7541

duke.contributor.orcid

Welsby, IJ|0000-0002-2789-5612

duke.contributor.orcid

Levy, JH|0000-0003-3766-4962

pubs.begin-page

115

pubs.end-page

122

pubs.issue

2

pubs.organisational-group

Duke

pubs.organisational-group

School of Medicine

pubs.organisational-group

Faculty

pubs.organisational-group

Clinical Science Departments

pubs.organisational-group

Anesthesiology

pubs.organisational-group

Anesthesiology, Cardiothoracic

pubs.organisational-group

Medicine

pubs.organisational-group

Surgery

pubs.organisational-group

Medicine, Hematology

pubs.organisational-group

Surgery, Cardiovascular and Thoracic Surgery

pubs.publication-status

Published

pubs.volume

9

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